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The Drug-Induced Respiratory Disease Website

Known since the 1940s (PMID 18883450). Comprehensive list of causal drugs and chemicals available at PMID 1564446. Methemoglobin is the oxidized (Fe3+) species of hemoglobin (Fe2+). Patients present with slate-grey cyanosis, low SpO2, normal SaO2 and PaO2. Normally, methemoglobin is <1%. Levels above 40% can be life-threatening, producing pulmonary edema, cardiovascular collapse (PMID 17122537) CNS disturbances and death. Management includes i.v. methylene blue. A possible rebound increase in MeHb upon treatment requires close monitoring. Excess methylene blue can also produce methemoglobinemia. Guidelines: PMID 34467556.

Publications

Hamza A, Nasrullah A, Singh R, DiSilvio B

Phenazopyridine-Induced Methaemoglobinaemia The Aftermath of Dysuria Treatment.

European journal of case reports in internal medicine 2022;9;003191 — 2022 — 003191

Murphy T, Fernandez M

Acquired methemoglobinemia from phenazopyridine use.

International journal of emergency medicine 2018 Nov 12;11;45 — 2018 Nov 12 — 45

Yu CH, Wang CH, Chang CC

Chocolate-colored blood with normal artery oxygen: methemoglobinemia related to phenazopyridine.

The American journal of the medical sciences 2011 Apr;341;337 — 2011 Apr — 337

Singh NK, Mirza N

Elderly woman with orange urine and purple hands.

Mayo Clinic proceedings 2008 Jul;83;744 — 2008 Jul — 744

Gold NA, Bithoney WG

Methemoglobinemia due to ingestion of at most three pills of pyridium in a 2-year-old: case report and review.

The Journal of emergency medicine 2003 Aug;25;143-8 — 2003 Aug — 143-8

Zimmerman RC, Green ED, Ghurabi WH, Colohan DP

Methemoglobinemia from overdose of phenazopyridine hydrochloride.

Annals of emergency medicine 1980 Mar;9;147-9 — 1980 Mar — 147-9

Jeffery WH, Zelicoff AP, Hardy WR

Acquired methemoglobinemia and hemolytic anemia after usual doses of phenazopyridine.

Drug intelligence & clinical pharmacy 1982 Feb;16;157-9 — 1982 Feb — 157-9